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Drug ReportsUsistapide
Usistapide
Usistapide is a small molecule pharmaceutical. It is currently being investigated in clinical studies.
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Clinical
Drug
Target
Variants
Financial
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Safety
Events Timeline
5D
1M
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6M
YTD
1Y
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5Y
Max
Events
FDA approval date
EMA approval date
Patent expiration date
Study first post date
Last update post date
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Completion date
Results first post date
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Commercial
Therapeutic Areas
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Trade Name
FDA
EMA
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Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
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Labels
FDA
EMA
Brand Name
Status
Last Update
10% methyl salicylate pain relief patchC2002632024-06-27
1st medxpatchunapproved drug other2026-01-08
365 whole foods market anticavity/antigingivitis mouthwashOTC monograph not final2022-05-12
5kind dmsoC2002632025-12-02
701 dieda zhengtong yaogao medicatedOTC monograph not final2019-11-13
701 dieda zhengtong yaogao medicated plasterOTC monograph not final2014-06-26
abejas y viboras roll onC2002632025-07-22
absolut skin spf 50 moisturizing sunscreenC2002632025-12-22
advanced antiseptic citrusC2002632025-02-20
advanced citrus antisepticC2002632025-01-10
Show 711 more
Indications
FDA
EMA
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Agency Specific
FDA
EMA
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Patent Expiration
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ATC Codes
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HCPCS
No data
Clinical
Clinical Trials
1805 clinical trials
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Indications Phases 4
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
AnesthesiaD0007587410283279
Healthy volunteers/patients57531579
Major depressive disorderD003865EFO_0003761F222416851061
NeoplasmsD009369C80321124955
Postoperative painD010149G89.18242172044
Emergence deliriumD000071257112162443
PainD010146EFO_0003843R52812431339
Prostatic neoplasmsD011471C6191962336
General anesthesiaD00076822591835
DeliriumD003693R41.0111131935
Show 285 more
Indications Phases 3
Indications Phases 2
Indications Phases 1
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Sleep wake disordersD012893G47246
AgingD000375GO_0007568R41.81145
Addictive behaviorD016739EFO_0004347314
Hepatic insufficiencyD04855033
Pick disease of the brainD020774EFO_0003096G31.01123
Hearing lossD034381EFO_0004238H91.9213
PharmacokineticsD01059933
Heart disease risk factorsD00008274233
VasoconstrictionD01466133
Migraine disordersD008881EFO_0003821G43213
Show 61 more
Indications Without Phase
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
SarcopeniaD055948EFO_1000653M62.8466
Dental plaqueD00377344
Urinary bladder neoplasmsD001749C6733
Deglutition disordersD003680R13.133
Brain ischemiaD002545EFO_0003883I67.8233
Trigger finger disorderD052582M65.333
Surgical blood lossD01606333
HypothermiaD007035T6833
Transurethral resection of prostateD02072822
Cerebral palsyD002547G8022
Show 231 more
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameUsistapide
INNusistapide
Description
Usistapide is a small molecule pharmaceutical. It is currently being investigated in clinical studies.
Classification
Small molecule
Drug classmicrosomal triglyceride transfer protein (MTP) inhibitors
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
COC(=O)[C@H](c1ccccc1)N1CCC(c2ccc(NC(=O)c3ccccc3-c3ccc(C(F)(F)F)cc3)cc2)CC1
Identifiers
PDB
CAS-ID403989-79-7
RxCUI
ChEMBL IDCHEMBL2103860
ChEBI ID
PubChem CID
DrugBank
UNII ID73YSY3U094 (ChemIDplus, GSRS)
Target
No data
Variants
No data
Financial
Revenue by drug
$
£
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Bloxiverz Avadel Pharmaceuticals
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Tabular view
Estimated US medical usage
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Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 753,244 documents
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Safety
Black-box Warning
Black-box warning for: Concerta, Cotempla xr-odt, Covaryx, Covaryx covaryx, Daytrana, Diclovix m, Dyural 40 kit, Dyural 80 kit, Dyural 80-lm, Dyural lm kit, Eemt, Eemt eemt, Esterified estrogens and methyltestosterone, Esterified estrogens and methyltestosterone full strength esterified estrogens and methyltestosterone half strength, Estratest f.s., Estratest f.s. estratest h.s., Estratest fs estratest hs, Fenovar, Healthy mamabe well rounded, Hydrocodone bitartrate and homatropine methylbromide, Hydromet, Jornay pm, Metadate cd, Metadate er, Methylene blue, Methylin, Methylphenidate, Methylphenidate hydrochloride, Methylphenidate hydrochloride (la), Methylphenidate hydrochloride cd, Methylphenidate hydrochloride extended release, Methylphenidate transdermal system, Orthaphen, Orthrexo, Perseris, Physicians ez use m-pred, Prenate elite, Prenate essential, Provayblue, Quillichew er, Quillivant, Relexxii, Ritalin, Torvex, Varophen
Adverse Events
Top Adverse Reactions
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244,367 adverse events reported
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