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Drug ReportsRegadenoson
Lexiscan, Rapiscan(regadenoson)
Lexiscan, Rapiscan, Regadenoson (regadenoson) is a small molecule pharmaceutical. Regadenoson was first approved as Lexiscan on 2008-04-10. It has been approved in Europe to treat myocardial perfusion imaging. The pharmaceutical is active against adenosine receptor A2a. In addition, it is known to target adenosine receptor A3, adenosine receptor A1, and adenosine receptor A2b.
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YTD
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FDA approval date
EMA approval date
Patent expiration date
Study first post date
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Commercial
Therapeutic Areas
Therapeutic Area
MeSH
diagnosisD003933
Trade Name
FDA
EMA
Lexiscan, Regadenoson
Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
Regadenoson
Tradename
Company
Number
Date
Products
LEXISCANAstellas PharmaN-022161 RX2008-04-10
1 products, RLD, RS
Labels
FDA
EMA
Brand Name
Status
Last Update
lexiscanNew Drug Application2018-12-21
lexiscan(r) (regadenoson)New Drug Application2024-01-28
regadenosonANDA2024-09-30
Indications
FDA
EMA
No data
Agency Specific
FDA
EMA
No data
Patent Expiration
Patent
Expires
Flag
FDA Information
Regadenoson, Lexiscan, Astellas
RE473012027-02-02DP
81061832027-02-02DP
ATC Codes
C: Cardiovascular system drugs
C01: Cardiac therapy drugs
C01E: Other cardiac preparations in atc
C01EB: Other plain cardiac preparations in atc
C01EB21: Regadenoson
HCPCS
Code
Description
J2785
Injection, regadenoson, 0.1 mg
Clinical
No data
Drug
General
Drug common nameRegadenoson
INNregadenoson
Description
Regadenoson is a purine nucleoside.
Classification
Small molecule
Drug classadenosine A receptor agonists
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
CNC(=O)c1cnn(-c2nc(N)c3ncn([C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O)c3n2)c1.O
Identifiers
PDB
CAS-ID313348-27-5
RxCUI1546015
ChEMBL IDCHEMBL3989695
ChEBI ID
PubChem CID219024
DrugBankDB06213
UNII ID7AXV542LZ4 (ChemIDplus, GSRS)
Target
Agency Approved
No data
Alternate
ADORA1
ADORA1
Organism
Homo sapiens
Gene name
ADORA1
Gene synonyms
NCBI Gene ID
Protein name
adenosine receptor A1
Protein synonyms
Uniprot ID
Mouse ortholog
Adora1 (11539)
adenosine receptor A1 (Q9WUF9)
Variants
No data
Financial
No data
Trends
No data
Safety
Black-box Warning
No Black-box warning
Adverse Events
0 adverse events reported
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