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Drug ReportsPexacerfont
Pexacerfont
Pexacerfont is a small molecule pharmaceutical. It is currently being investigated in clinical studies. It is known to target CRHR1-IT1-CRHR1 protein.
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Commercial
Clinical
Drug
Target
Variants
Financial
Trends
Safety
Events Timeline
5D
1M
3M
6M
YTD
1Y
2Y
5Y
Max
Events
FDA approval date
EMA approval date
Patent expiration date
Study first post date
Last update post date
Start date
Primary completion date
Completion date
Results first post date
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Commercial
No data
Clinical
Clinical Trials
12 clinical trials
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Indications Phases 4
No data
Indications Phases 3
No data
Indications Phases 2
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Irritable bowel syndromeD043183EFO_0000555K5811———2
Indications Phases 1
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
SyndromeD013577——1————1
Indications Without Phase
No data
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common namePexacerfont
INNpexacerfont
Description
Pexacerfont is a pyrazolopyridine.
Classification
Small molecule
Drug classCRF-1 (corticotropin releasing factor) receptor antagonists
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
CC[C@@H](C)Nc1nc(C)nc2c(-c3ccc(OC)nc3C)c(C)nn12
Identifiers
PDB—
CAS-ID459856-18-9
RxCUI—
ChEMBL IDCHEMBL482950
ChEBI ID—
PubChem CID9884366
DrugBankDB12572
UNII IDLF1VBG4ZUK (ChemIDplus, GSRS)
Target
Agency Approved
No data
Alternate
LINC02210-CRHR1
LINC02210-CRHR1
Organism
Homo sapiens
Gene name
LINC02210-CRHR1
Gene synonyms
CRFR, CRFR1, CRHR
NCBI Gene ID
104909134
Protein name
CRHR1-IT1-CRHR1 protein
Protein synonyms
Corticotropin-releasing hormone receptor 1, CRH-R-1, CRH-R1, CRHR1-IT1-CRHR1 readthrough
Uniprot ID
B4DMR5
Mouse ortholog
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Variants
No data
Financial
No data
Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 668 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
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1 adverse events reported
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