Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
---|---|---|---|---|---|---|---|---|---|
Neoplasms | D009369 | — | C80 | 2 | 1 | 1 | — | — | 3 |
Essential thrombocythemia | D013920 | — | D47.3 | 1 | 1 | 1 | — | — | 2 |
Primary myelofibrosis | D055728 | — | D47.4 | 1 | 1 | 1 | — | — | 2 |
Thrombocytosis | D013922 | — | D75.83 | 1 | 1 | 1 | — | — | 2 |
Hematologic neoplasms | D019337 | — | — | 1 | — | 1 | — | — | 2 |
Polycythemia vera | D011087 | — | D45 | — | — | 1 | — | — | 1 |
Polycythemia | D011086 | EFO_0005804 | D75.1 | — | — | 1 | — | — | 1 |
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
---|---|---|---|---|---|---|---|---|---|
Leukemia | D007938 | — | C95 | 1 | 1 | — | — | — | 1 |
Myelodysplastic syndromes | D009190 | — | D46 | 1 | 1 | — | — | — | 1 |
Myeloid leukemia acute | D015470 | — | C92.0 | 1 | 1 | — | — | — | 1 |
Myeloproliferative disorders | D009196 | — | D47.1 | 1 | 1 | — | — | — | 1 |
Hematologic diseases | D006402 | EFO_0005803 | D75.9 | 1 | 1 | — | — | — | 1 |
Precancerous conditions | D011230 | — | — | 1 | 1 | — | — | — | 1 |
Myelodysplastic-myeloproliferative diseases | D054437 | — | — | 1 | 1 | — | — | — | 1 |
Myeloid leukemia | D007951 | — | C92 | 1 | 1 | — | — | — | 1 |
Preleukemia | D011289 | — | — | 1 | 1 | — | — | — | 1 |
Bone marrow diseases | D001855 | — | — | 1 | 1 | — | — | — | 1 |
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
---|---|---|---|---|---|---|---|---|---|
Multiple myeloma | D009101 | — | C90.0 | 1 | — | — | — | — | 1 |
Plasma cell neoplasms | D054219 | — | — | 1 | — | — | — | — | 1 |
Lymphoma | D008223 | — | C85.9 | 1 | — | — | — | — | 1 |
Drug common name | Pelabresib |
INN | pelabresib |
Description | Pelabresib is a small molecule pharmaceutical. It is currently being investigated in clinical studies. It is known to target bromodomain-containing protein 4. |
Classification | Small molecule |
Drug class | extra-terminal motif (BET) family of bromodomain (BRD) proteins |
Image (chem structure or protein) | ![]() |
Structure (InChI/SMILES or Protein Sequence) | Cc1noc2c1-c1ccccc1C(c1ccc(Cl)cc1)=N[C@H]2CC(N)=O |
PDB | — |
CAS-ID | 1380087-89-7 |
RxCUI | — |
ChEMBL ID | CHEMBL4303404 |
ChEBI ID | — |
PubChem CID | 57389999 |
DrugBank | DB17129 |
UNII ID | U4017GUQ06 (ChemIDplus, GSRS) |