Enzastaurin
Enzastaurin is a small molecule pharmaceutical. It is currently being investigated in clinical studies. The pharmaceutical is active against protein kinase C beta type. In addition, it is known to target protein kinase C alpha type, protein kinase C delta type, and protein kinase C gamma type.
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Commercial
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Clinical
Clinical Trials
51 clinical trials
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Indications Phases 4
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Indications Phases 3
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Indications Phases 2
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Colorectal neoplasms | D015179 | — | — | — | 1 | — | — | — | 1 |
Indications Phases 1
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Indications Without Phase
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Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
| Drug common name | Enzastaurin |
| INN | enzastaurin |
| Description | 3-(1-methyl-3-indolyl)-4-[1-[1-(2-pyridinylmethyl)-4-piperidinyl]-3-indolyl]pyrrole-2,5-dione is a member of indoles and a member of maleimides. |
| Classification | Small molecule |
| Drug class | — |
| Image (chem structure or protein) |  |
| Structure (InChI/SMILES or Protein Sequence) | Cn1cc(C2=C(c3cn(C4CCN(Cc5ccccn5)CC4)c4ccccc34)C(=O)NC2=O)c2ccccc21 |
Identifiers
| PDB | — |
| CAS-ID | 170364-57-5 |
| RxCUI | — |
| ChEMBL ID | CHEMBL300138 |
| ChEBI ID | — |
| PubChem CID | 176167 |
| DrugBank | — |
| UNII ID | UC96G28EQF (ChemIDplus, GSRS) |
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Safety
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Adverse Events
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261 adverse events reported
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