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AboutPricing
Drug ReportsCyproterone
Cyproterone acetate
Cyproterone acetate is a small molecule pharmaceutical. It is currently being investigated in clinical studies. The pharmaceutical is active against androgen receptor.
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Events Timeline
5D
1M
3M
6M
YTD
1Y
2Y
5Y
Max
Events
FDA approval date
EMA approval date
Patent expiration date
Study first post date
Last update post date
Start date
Primary completion date
Completion date
Results first post date
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Commercial
Therapeutic Areas
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Trade Name
FDA
EMA
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Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
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Labels
FDA
EMA
Brand Name
Status
Last Update
dianeal low calcium peritoneal dialysis solution with dextrose dianeal pd-2 peritoneal dialysis solution with dextroseNew Drug Application2013-06-30
dianeal low calcium with dextroseunapproved drug for use in drug shortage2025-03-17
dianeal low calcium with dextrose dianeal pd-2 with dextroseunapproved drug for use in drug shortage2025-03-10
dianeal pd-2 peritoneal dialysis solution with dextroseNew Drug Application2010-06-07
dianeal pd-2 with dextroseunapproved drug for use in drug shortage2025-03-10
emme diane pure protection tinted antioxidant sunscreenC2002632025-01-16
emme diane tinted mineral sunscreenC2002632025-01-16
Indications
FDA
EMA
No data
Agency Specific
FDA
EMA
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Patent Expiration
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ATC Codes
G: Genito urinary system and sex hormones
— G03: Sex hormones and modulators of the genital system
— G03H: Antiandrogen sex hormones and modulators of the genital system
— G03HA: Antiandrogens, plain
— G03HA01: Cyproterone
— G03HB: Antiandrogens and estrogens
— G03HB01: Cyproterone and estrogen
HCPCS
No data
Clinical
Clinical Trials
61 clinical trials
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Indications Phases 4
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Indications Phases 3
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Acne vulgarisD000152EFO_0003894L70——1—23
Indications Phases 2
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Indications Phases 1
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Indications Without Phase
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Prostatic neoplasmsD011471—C61————44
AlopeciaD000505—L64————22
Seborrheic dermatitisD012628—L21————22
HirsutismD006628—L68.0————22
AnemiaD000740EFO_0004272D64.9————11
Erectile dysfunctionD007172EFO_0004234F52.21————11
VirilismD014770——————11
HypersensitivityD006967EFO_0003785T78.40————11
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameCyproterone acetate
INNcyproterone
Description
Cyproterone acetate is a steroid ester resulting from the formal condensation of the carboxy group of acetic acid with the 17-hydroxy group of cyproterone. It is an antiandrogenic drug which has recently been recognized to promote the occurrence and growth of intracranial meningiomas. It has a role as an androgen antagonist, a progestin and a geroprotector. It is a 20-oxo steroid, a 3-oxo-Delta(4) steroid, a chlorinated steroid, a steroid ester and an acetate ester. It is functionally related to a cyproterone.
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Classification
Small molecule
Drug classantiandrogens
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
CC(=O)O[C@]1(C(C)=O)CC[C@H]2[C@@H]3C=C(Cl)C4=CC(=O)[C@@H]5C[C@@H]5[C@]4(C)[C@H]3CC[C@@]21C
Identifiers
PDB—
CAS-ID427-51-0
RxCUI—
ChEMBL IDCHEMBL139835
ChEBI ID50743
PubChem CID9880
DrugBankDB04839
UNII IDE61Q31EK2F (ChemIDplus, GSRS)
Target
Agency Approved
AR
AR
Organism
Homo sapiens
Gene name
AR
Gene synonyms
DHTR, NR3C4
NCBI Gene ID
367
Protein name
androgen receptor
Protein synonyms
Dihydrotestosterone receptor, Nuclear receptor subfamily 3 group C member 4
Uniprot ID
Q9UD95
Mouse ortholog
Ar (11835)
androgen receptor (P19091)
Alternate
No data
Variants
No data
Financial
No data
Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 43,591 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
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147,633 adverse events reported
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