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Drug ReportsBilastine
Bilastine
Bilastine is a small molecule pharmaceutical. It is currently being investigated in clinical studies. It is known to target histamine H1 receptor.
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Variants
Financial
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Events Timeline
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YTD
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5Y
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Events
FDA approval date
EMA approval date
Patent expiration date
Study first post date
Last update post date
Start date
Primary completion date
Completion date
Results first post date
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Commercial
Therapeutic Areas
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Trade Name
FDA
EMA
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Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
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Labels
FDA
EMA
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Indications
FDA
EMA
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Agency Specific
FDA
EMA
No data
Patent Expiration
No data
ATC Codes
R: Respiratory system drugs
— R06: Antihistamines for systemic use
— R06A: Antihistamines for systemic use
— R06AX: Other antihistamines for systemic use in atc
— R06AX29: Bilastine
S: Sensory organ drugs
— S01: Ophthalmologicals
— S01G: Decongestants and antiallergics
— S01GX: Other antiallergics in atc
— S01GX13: Bilastine
HCPCS
No data
Clinical
Clinical Trials
25 clinical trials
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Indications Phases 4
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Allergic rhinitisD065631—J30.9—343—10
RhinitisD012220EFO_0008521J31—343—10
UrticariaD014581EFO_0005531L501332—7
Allergic rhinitis seasonalD006255EFO_0003956J30—331—7
Allergic conjunctivitisD003233EFO_0007141H10.441321—6
AsthmaD001249EFO_0000270J45———1—1
Indications Phases 3
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
ConjunctivitisD003231HP_0000509H10132——5
Chronic urticariaD000080223—L50.8122——4
Allergic rhinitis perennialD012221EFO_1001417J30.89——1——1
Indications Phases 2
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
HypersensitivityD006967HP_0012393T78.40—1———1
Indications Phases 1
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Healthy volunteers/patients———4————4
PharmacokineticsD010599——1————1
Indications Without Phase
No data
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameBilastine
INNbilastine
Description
Bilastine is a member of benzimidazoles.
Classification
Small molecule
Drug classantihistaminics (histamine-H1 receptor antagonists)
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
CCOCCn1c(C2CCN(CCc3ccc(C(C)(C)C(=O)O)cc3)CC2)nc2ccccc21
Identifiers
PDB—
CAS-ID202189-78-4
RxCUI—
ChEMBL IDCHEMBL1742423
ChEBI ID—
PubChem CID185460
DrugBankDB11591
UNII IDPA1123N395 (ChemIDplus, GSRS)
Target
Agency Approved
No data
Alternate
HRH1
HRH1
Organism
Homo sapiens
Gene name
HRH1
Gene synonyms
NCBI Gene ID
Protein name
histamine H1 receptor
Protein synonyms
histamine receptor, subclass H1
Uniprot ID
Mouse ortholog
Hrh1 (15465)
histamine H1 receptor (Q91XN3)
Variants
No data
Financial
No data
Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 442 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
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647 adverse events reported
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