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Drug ReportsBenzocaine
Benzocaine
Benzocaine is a small molecule pharmaceutical. It is currently being investigated in clinical studies.
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Events Timeline
5D
1M
3M
6M
YTD
1Y
2Y
5Y
Max
Events
FDA approval date
EMA approval date
Patent expiration date
Study first post date
Last update post date
Start date
Primary completion date
Completion date
Results first post date
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Commercial
Therapeutic Areas
Therapeutic Area
MeSH
infectionsD007239
digestive system diseasesD004066
stomatognathic diseasesD009057
otorhinolaryngologic diseasesD010038
cardiovascular diseasesD002318
skin and connective tissue diseasesD017437
signs and symptoms pathological conditionsD013568
wounds and injuriesD014947
Trade Name
FDA
EMA
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Drug Products
FDA
EMA
New Drug Application (NDA)
New Drug Application (NDA)
Abbreviated New Drug Application (ANDA)
Abbreviated New Drug Application (ANDA)
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Labels
FDA
EMA
Brand Name
Status
Last Update
10 person ansiOTC monograph final2010-06-07
20/20OTC monograph final2012-05-08
25 person ansiOTC monograph final2010-06-07
2x med liqOTC monograph not final2021-09-02
3x medicated mouth sore gelC2002632025-07-22
3x medicated toothache and gum gelC2002632025-01-20
4x medicated gum creamC2002632025-03-12
4x medicated severe toothache and gum creamC2002632025-01-19
4x medicated severe toothache and gum gelC2002632025-01-19
4x medicated toothache and gum creamC2002632025-04-11
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Indications
FDA
EMA
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Agency Specific
FDA
EMA
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Patent Expiration
No data
ATC Codes
C: Cardiovascular system drugs
C05: Vasoprotectives
C05A: Agents for treatment of hemorrhoids and anal fissures for topical use
C05AD: Local anesthetics for treatment of hemorrhoids and anal fissures for topical use
C05AD03: Benzocaine
D: Dermatologicals
D04: Antipruritics, incl. antihistamines, anesthetics, etc.
D04A: Antipruritics, incl. antihistamines, anesthetics, etc.
D04AB: Anesthetics for topical use
D04AB04: Benzocaine
N: Nervous system drugs
N01: Anesthetics
N01B: Local anesthetics
N01BA: Esters of aminobenzoic acid for local anesthesia
N01BA05: Benzocaine
R: Respiratory system drugs
R02: Throat preparations
R02A: Throat preparations
R02AD: Local anesthetic throat preparations
R02AD01: Benzocaine
HCPCS
No data
Clinical
Clinical Trials
6482 clinical trials
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Indications Phases 4
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Indications Phases 3
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Indications Phases 2
Indication
MeSH
Ontology
ICD-10
Ph 1
Ph 2
Ph 3
Ph 4
Other
Total
Stress fracturesD015775M84.311
Post-traumatic stress disordersD013313EFO_0001358F43.111
Traumatic stress disorders acuteD040701EFO_0005223F43.011
Indications Phases 1
No data
Indications Without Phase
No data
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
Drug common nameBenzocaine
INNbenzocaine
Description
Benzocaine is a benzoate ester having 4-aminobenzoic acid as the acid component and ethanol as the alcohol component. A surface anaesthetic, it is used to suppress the gag reflex, and as a lubricant and topical anaesthetic on the larynx, mouth, nasal cavity, respiratory tract, oesophagus, rectum, urinary tract, and vagina. It has a role as a topical anaesthetic, an antipruritic drug, an allergen and a sensitiser. It is a benzoate ester and a substituted aniline.
Classification
Small molecule
Drug classlocal anesthetics
Image (chem structure or protein)Loading
Structure (InChI/SMILES or Protein Sequence)
CCOC(=O)c1ccc(N)cc1
Identifiers
PDB
CAS-ID94-09-7
RxCUI
ChEMBL IDCHEMBL278172
ChEBI ID116735
PubChem CID2337
DrugBankDB01086
UNII IDU3RSY48JW5 (ChemIDplus, GSRS)
Target
No data
Variants
No data
Financial
Revenue by drug
$
£
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Estimated US medical usage
Benzocaine
Total medical expenditures per year (USD, in millions)
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Benzocaine
+
Menthol
Total medical expenditures per year (USD, in millions)
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Benzocaine
+
Trimethobenzamide
Total medical expenditures per year (USD, in millions)
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Tabular view
Trends
PubMed Central
Top Terms for Disease or Syndrome:
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Additional graphs summarizing 249,527 documents
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Safety
Black-box Warning
No Black-box warning
Adverse Events
Top Adverse Reactions
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305,048 adverse events reported
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