Benzocaine
Benzocaine is a small molecule pharmaceutical. It is currently being investigated in clinical studies.
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Events Timeline
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Commercial
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Drug Products
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New Drug Application (NDA)
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Abbreviated New Drug Application (ANDA)
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Labels
FDA
EMA
Brand Name | Status | Last Update |
|---|---|---|
| 20/20 | OTC monograph final | 2012-05-08 |
| 2x med liq | OTC monograph not final | 2021-09-02 |
| 3x medicated mouth sore gel | C200263 | 2025-01-20 |
| 3x medicated toothache and gum gel | C200263 | 2025-01-20 |
| 4x medicated gum cream | C200263 | 2025-03-12 |
| 4x medicated severe toothache and gum cream | C200263 | 2025-01-19 |
| 4x medicated severe toothache and gum gel | C200263 | 2025-01-19 |
| 4x medicated toothache and gum cream | C200263 | 2025-04-11 |
| 4x medicated toothache and gum gel | C200263 | 2025-01-20 |
| 7 select oral pain maximum strength relief | C200263 | 2024-12-02 |
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Indications
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Agency Specific
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Patent Expiration
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ATC Codes
C: Cardiovascular system drugs
— C05: Vasoprotectives
— C05A: Agents for treatment of hemorrhoids and anal fissures for topical use
— C05AD: Local anesthetics for treatment of hemorrhoids and anal fissures for topical use
— C05AD03: Benzocaine
D: Dermatologicals
— D04: Antipruritics, incl. antihistamines, anesthetics, etc.
— D04A: Antipruritics, incl. antihistamines, anesthetics, etc.
— D04AB: Anesthetics for topical use
— D04AB04: Benzocaine
N: Nervous system drugs
— N01: Anesthetics
— N01B: Local anesthetics
— N01BA: Esters of aminobenzoic acid for local anesthesia
— N01BA05: Benzocaine
R: Respiratory system drugs
— R02: Throat preparations
— R02A: Throat preparations
— R02AD: Local anesthetic throat preparations
— R02AD01: Benzocaine
HCPCS
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Clinical
Clinical Trials
6366 clinical trials
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Indications Phases 4
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Neuromuscular blockade | D019148 | — | — | — | — | 1 | 3 | — | 4 |
| Prostatic neoplasms | D011471 | — | C61 | — | 2 | — | 1 | — | 3 |
| Anesthesia | D000758 | — | — | — | — | 2 | 1 | — | 3 |
| Acute coronary syndrome | D054058 | EFO_0005672 | — | — | — | — | 1 | — | 1 |
| Chronic renal insufficiency | D051436 | — | N18 | — | — | — | 1 | — | 1 |
| Kidney diseases | D007674 | EFO_0003086 | N08 | — | — | — | 1 | — | 1 |
| Leiomyoma | D007889 | — | D25 | — | — | — | 1 | — | 1 |
| Endometriosis | D004715 | EFO_0001065 | N80 | — | — | — | 1 | — | 1 |
| Cholecystitis | D002764 | — | K81 | — | — | — | 1 | — | 1 |
| Uterine prolapse | D014596 | EFO_1001864 | N81.4 | — | — | — | 1 | — | 1 |
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Indications Phases 3
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Diabetes mellitus | D003920 | EFO_0000400 | E08-E13 | 4 | — | 1 | — | 1 | 6 |
| Hepatitis c | D006526 | — | B19.2 | — | 4 | 1 | — | — | 5 |
| Hepatitis | D006505 | — | K75.9 | — | 4 | 1 | — | — | 5 |
| Chronic hepatitis c | D019698 | EFO_0004220 | B18.2 | — | 3 | 1 | — | — | 4 |
| Hepatitis a | D006506 | EFO_0007305 | B15 | — | 3 | 1 | — | — | 4 |
| Hiv infections | D015658 | EFO_0000764 | B20 | — | 1 | 1 | — | — | 2 |
| Acquired immunodeficiency syndrome | D000163 | EFO_0000765 | B20 | — | — | 1 | — | — | 1 |
| Hiv-2 | D015498 | — | — | — | — | 1 | — | — | 1 |
| Immunologic deficiency syndromes | D007153 | — | D84.9 | — | — | 1 | — | — | 1 |
| Small cell lung carcinoma | D055752 | — | — | — | — | 1 | — | — | 1 |
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Indications Phases 2
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Chronic hepatitis | D006521 | — | K73.9 | — | 1 | — | — | — | 1 |
| Liver cirrhosis | D008103 | EFO_0001422 | K74.0 | — | 1 | — | — | — | 1 |
| Fibrosis | D005355 | — | — | — | 1 | — | — | — | 1 |
| Hiv | D006678 | — | O98.7 | — | 1 | — | — | — | 1 |
| Castration-resistant prostatic neoplasms | D064129 | — | — | — | 1 | — | — | — | 1 |
| Non-small-cell lung carcinoma | D002289 | — | — | — | 1 | — | — | — | 1 |
| Lung neoplasms | D008175 | — | C34.90 | — | 1 | — | — | — | 1 |
| Alzheimer disease | D000544 | EFO_0000249 | F03 | — | 1 | — | — | — | 1 |
| Dementia | D003704 | EFO_0003862 | F03 | — | 1 | — | — | — | 1 |
| Thyroid neoplasms | D013964 | EFO_0003841 | — | — | 1 | — | — | — | 1 |
Show 1 more
Indications Phases 1
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Type 1 diabetes mellitus | D003922 | EFO_0001359 | E10 | 3 | — | — | — | — | 3 |
| Type 2 diabetes mellitus | D003924 | EFO_0001360 | E11 | 3 | — | — | — | — | 3 |
| Hypoglycemia | D007003 | — | E16.2 | 1 | — | — | — | — | 1 |
Indications Without Phase
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Postoperative complications | D011183 | — | — | — | — | — | — | 1 | 1 |
| Pneumonia | D011014 | EFO_0003106 | J18 | — | — | — | — | 1 | 1 |
| Wound infection | D014946 | — | — | — | — | — | — | 1 | 1 |
| Surgical wound infection | D013530 | — | — | — | — | — | — | 1 | 1 |
Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
| Drug common name | Benzocaine |
| INN | benzocaine |
| Description | Benzocaine is a benzoate ester having 4-aminobenzoic acid as the acid component and ethanol as the alcohol component. A surface anaesthetic, it is used to suppress the gag reflex, and as a lubricant and topical anaesthetic on the larynx, mouth, nasal cavity, respiratory tract, oesophagus, rectum, urinary tract, and vagina. It has a role as a topical anaesthetic, an antipruritic drug, an allergen and a sensitiser. It is a benzoate ester and a substituted aniline. |
| Classification | Small molecule |
| Drug class | local anesthetics |
| Image (chem structure or protein) |  |
| Structure (InChI/SMILES or Protein Sequence) | CCOC(=O)c1ccc(N)cc1 |
Identifiers
| PDB | — |
| CAS-ID | 94-09-7 |
| RxCUI | — |
| ChEMBL ID | CHEMBL278172 |
| ChEBI ID | 116735 |
| PubChem CID | 2337 |
| DrugBank | DB01086 |
| UNII ID | U3RSY48JW5 (ChemIDplus, GSRS) |
Target
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Variants
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Financial
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Estimated US medical usage
Benzocaine
Total medical expenditures per year (USD, in millions)
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Benzocaine
+
Menthol
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Benzocaine
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Trimethobenzamide
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Trends
PubMed Central
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Additional graphs summarizing 245,070 documents
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Safety
Black-box Warning
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Adverse Events
Top Adverse Reactions
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305,048 adverse events reported
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