BURAPITANT
Burapitant is a small molecule pharmaceutical. It is currently being investigated in clinical studies.
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Commercial
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Clinical
Clinical Trials
2 clinical trials
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Indications Phases 4
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Indications Phases 3
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Indications Phases 2
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Overactive urinary bladder | D053201 | EFO_1000781 | N32.81 | — | 2 | — | — | — | 2 |
| Urge urinary incontinence | D053202 | EFO_0006865 | N39.41 | — | 1 | — | — | — | 1 |
| Urinary incontinence | D014549 | HP_0000020 | R32 | — | 1 | — | — | — | 1 |
| Enuresis | D004775 | — | R32 | — | 1 | — | — | — | 1 |
Indications Phases 1
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Indications Without Phase
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Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
| Drug common name | BURAPITANT |
| INN | burapitant |
| Description | Burapitant (SSR-240,600) is a drug developed by Sanofi-Aventis which was one of the first compounds developed that acts as a potent and selective antagonist for the NK1 receptor. While burapitant itself did not proceed beyond early clinical trials and was never developed for clinical use in humans, promising animal results from this and related compounds have led to a number of novel drugs from this class that have now been introduced into medical use.
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| Classification | Small molecule |
| Drug class | tachykinin (neurokinin) receptor antagonists: NK1 receptor antagonists |
| Image (chem structure or protein) |  |
| Structure (InChI/SMILES or Protein Sequence) | CC(C)(C(N)=O)C1CCN(CCC2(c3ccc(Cl)c(Cl)c3)CN(C(=O)Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)CCO2)CC1 |
Identifiers
| PDB | — |
| CAS-ID | 537034-22-3 |
| RxCUI | — |
| ChEMBL ID | CHEMBL3544947 |
| ChEBI ID | — |
| PubChem CID | 23649599 |
| DrugBank | — |
| UNII ID | E35SK332MS (ChemIDplus, GSRS) |
Target
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Financial
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Trends
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Safety
Black-box Warning
No Black-box warning
Adverse Events
0 adverse events reported
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