Azatadine
Optimine, Trinalin (azatadine) is a small molecule pharmaceutical. Azatadine was first approved as Optimine on 1982-01-01. It is used to treat allergic rhinitis perennial, allergic rhinitis seasonal, ear diseases, respiration disorders, and urticaria in the USA.
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Azatadine maleate
Tradename | Company | Number | Date | Products |
|---|---|---|---|---|
| OPTIMINE | Merck & Co | N-017601 DISCN | 1982-01-01 | 1 products |
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Azatadine maleate
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Pseudoephedrine sulfate
Tradename | Company | Number | Date | Products |
|---|---|---|---|---|
| TRINALIN | Merck & Co | N-018506 DISCN | 1982-03-23 | 1 products |
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General
| Drug common name | Azatadine |
| INN | azatadine |
| Description | Azatadine is a benzo[5,6]cyclohepta[1,2-b]pyridine having a 1-methylpiperidin-4-ylidene group at the 11-position. It has a role as a H1-receptor antagonist and an anti-allergic agent. It is a benzocycloheptapyridine and a tertiary amine. |
| Classification | Small molecule |
| Drug class | tricyclic histaminic-H1 receptor antagonists, loratadine derivatives (formerly-tadine) |
| Image (chem structure or protein) |  |
| Structure (InChI/SMILES or Protein Sequence) | CN1CCC(=C2c3ccccc3CCc3cccnc32)CC1 |
Identifiers
| PDB | — |
| CAS-ID | 3964-81-6 |
| RxCUI | — |
| ChEMBL ID | CHEMBL946 |
| ChEBI ID | 2946 |
| PubChem CID | 19861 |
| DrugBank | DB00719 |
| UNII ID | 94Z39NID6C (ChemIDplus, GSRS) |
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Azatadine
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Azatadine
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Pseudoephedrine
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17 adverse events reported
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