Antazoline
Vasocon-a (antazoline) is a small molecule pharmaceutical. Antazoline was first approved as Vasocon-a on 1994-07-11. It is used to treat allergic conjunctivitis, pruritus, and respiration disorders in the USA.
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ATC Codes
R: Respiratory system drugs
— R01: Nasal preparations
— R01A: Decongestants and other nasal preparations for topical use
— R01AC: Antiallergic nasal preparations for topical use, excl. corticosteroids
— R01AC04: Antazoline
— R06: Antihistamines for systemic use
— R06A: Antihistamines for systemic use
— R06AX: Other antihistamines for systemic use in atc
— R06AX05: Antazoline
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Clinical
Clinical Trials
10 clinical trials
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Indications Phases 4
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Atrial fibrillation | D001281 | EFO_0000275 | I48.0 | — | — | — | 2 | 1 | 3 |
| Allergic conjunctivitis | D003233 | EFO_0007141 | H10.44 | — | — | 2 | 1 | — | 3 |
| Conjunctivitis | D003231 | — | H10 | — | — | — | 1 | — | 1 |
Indications Phases 3
Indication | MeSH | Ontology | ICD-10 | Ph 1 | Ph 2 | Ph 3 | Ph 4 | Other | Total |
|---|---|---|---|---|---|---|---|---|---|
| Pterygium | D011625 | — | H11.0 | — | — | 1 | — | — | 1 |
| Inflammation | D007249 | MP_0001845 | — | — | — | 1 | — | — | 1 |
| Respiration disorders | D012120 | — | J00-J99 | — | — | 1 | — | — | 1 |
| Hypersensitivity | D006967 | EFO_0003785 | T78.40 | — | — | 1 | — | — | 1 |
| Cold temperature | D003080 | — | — | — | — | 1 | — | — | 1 |
Indications Phases 2
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Epidemiology
Epidemiological information for investigational and approved indications
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Drug
General
| Drug common name | Antazoline |
| INN | antazoline |
| Description | Antazoline is a member of the class of imidazolines that is 2-aminomethyl-2-imidazoline in which the exocyclic amino hydrogens are replaced by benzyl and phenyl groups. Antazoline is only found in individuals that have taken the drug. It has a role as a H1-receptor antagonist, a cholinergic antagonist and a xenobiotic. It is a tertiary amino compound, an aromatic amine and a member of imidazolines. |
| Classification | Small molecule |
| Drug class | antihistamines/local vasoconstrictors (antazoline type) |
| Image (chem structure or protein) |  |
| Structure (InChI/SMILES or Protein Sequence) | c1ccc(CN(CC2=NCCN2)c2ccccc2)cc1 |
Identifiers
| PDB | — |
| CAS-ID | 91-75-8 |
| RxCUI | — |
| ChEMBL ID | CHEMBL1305 |
| ChEBI ID | 84115 |
| PubChem CID | 2200 |
| DrugBank | DB08799 |
| UNII ID | DHA8014SS1 (ChemIDplus, GSRS) |
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Antazoline
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Naphazoline
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